Orlistat — Clinical Evidence

All published trials referenced on this site. Click any source link to read the original journal article.

Last reviewed: March 2026

Medical disclaimer: This website is for informational purposes only and does not constitute medical advice. Always consult a qualified healthcare provider before starting, stopping, or changing any treatment.

Randomised controlled trials

In the following trials, participants were randomly assigned to Orlistat or a dummy pill (placebo). All weight loss figures are average body weight reductions from baseline.

TrialKey resultSource
[1]XENDOS2.8 kg more weight loss than placebo at 4 years. 37% reduction in progression to type 2 diabetes vs. placebo plus lifestyle intervention.Diabetes Care 2004
[2]1-year randomised controlled trial (Sjöström et al.)8.5% average weight loss in the orlistat group vs 5.4% placebo — the most commonly cited 1-year efficacy figure. The drug's effect is modest compared to GLP-1 class drugs but it works through a completely different mechanism (blocking fat absorption in the gut, not the brain).International Journal of Obesity 2000

Reported side effects

Frequencies from XENDOS. View source ↗

Side effectFrequency in trial
Oily/fatty stools (steatorrhoea)
27%
Faecal urgency
22%
Oily spotting on underwear
27%
Faecal incontinence
8%
Abdominal pain/discomfort
14%

Body composition data

No specific body composition data distinguishes orlistat from calorie-restriction alone. The drug produces weight loss entirely through calorie malabsorption — lean mass effects depend on the degree of calorie deficit and protein intake.

Cardiovascular & metabolic data

In the 4-year XENDOS trial, orlistat reduced progression from prediabetes to type 2 diabetes by 37% compared to placebo plus lifestyle changes. Modest improvements in blood pressure and LDL observed.